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Assay Detail

CHEMBL5584834

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of FGFR1 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Fibroblast growth factor receptor 1 (CHEMBL3650)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Recent advances in c-Met-based dual inhibitors in the treatment of cancers.
Jin F, Lin Y, Yuan W, Wu S, Yang M, Ding S, Liu J, Chen Y.
Eur J Med Chem (2024) 272 : 116477 -116477
PubMed 38733884 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.75 7.75

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3808948 1 7.75

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3808948 IC50 = 18.0 nM 7.75