Assay Detail
Binding
CHEMBL5620541
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of full length PDE7 (unknown origin) using FAM-cAMP as substrate by fluorescence based analysis
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Advances in the development of phosphodiesterase 7 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 6.69 | 8.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5625053 | — | — | 1 | 8.26 |
| CHEMBL5630856 | — | — | 1 | 8.21 |
| CHEMBL5624926 | — | — | 1 | 7.70 |
| CHEMBL183965 | — | — | 1 | 7.26 |
| CHEMBL5624721 | — | — | 1 | 7.13 |
| CHEMBL5625128 | — | — | 1 | 7.00 |
| CHEMBL5629944 | — | — | 1 | 6.89 |
| CHEMBL1236215 | — | — | 1 | 6.29 |
| CHEMBL1927722 | — | — | 1 | 6.26 |
| CHEMBL3545918 | — | — | 1 | 5.96 |
| CHEMBL5630770 | — | — | 1 | 5.94 |
| CHEMBL184334 | — | — | 1 | 5.82 |
| CHEMBL5631032 | — | — | 1 | 5.80 |
| CHEMBL503420 | — | — | 1 | 5.10 |
| CHEMBL5625119 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5625053 | — | IC50 | = | 5.5 | nM | 8.26 |
| CHEMBL5630856 | — | IC50 | = | 6.1 | nM | 8.21 |
| CHEMBL5624926 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL183965 | — | IC50 | = | 55.0 | nM | 7.26 |
| CHEMBL5624721 | — | IC50 | = | 74.0 | nM | 7.13 |
| CHEMBL5625128 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL5629944 | — | IC50 | = | 130.0 | nM | 6.89 |
| CHEMBL1236215 | — | IC50 | = | 510.0 | nM | 6.29 |
| CHEMBL1927722 | — | IC50 | = | 550.0 | nM | 6.26 |
| CHEMBL3545918 | — | IC50 | = | 1110.0 | nM | 5.96 |
| CHEMBL5630770 | — | IC50 | = | 1150.0 | nM | 5.94 |
| CHEMBL184334 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL5631032 | — | IC50 | = | 1590.0 | nM | 5.80 |
| CHEMBL503420 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL5625119 | — | IC50 | < | 10.0 | nM | - |