Assay Detail
Binding
CHEMBL5724014
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NanoLuc NanoBRET (CIT)
2
Total Activities
2
Compounds Tested
1
Activity Types
2
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Data for DCP probe C3TD879
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 8.02 | 8.02 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Target protein length | Target protein length | - | — | full length |
| Target protein type | Target protein type | - | — | Implied Kd values calculated using Tracer K10 Kd = 230 nM; Tracer K10 used at 1 µM for CITK NanoBRET |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5572737 | — | — | 1 | 8.02 |
| CHEMBL5571434 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5572737 | — | Kd | = | 9.5 | nM | 8.02 |
| CHEMBL5571434 | — | Kd | = | - | — | - |