Assay Detail
Binding
CHEMBL617470
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Ability to displace [3H]ketanserin from rat cortical homogenate 5-hydroxytryptamine 2A receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Dihydrobenzofuran analogues of hallucinogens. 4. Mescaline derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.47 | 5.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL319415 | — | — | 1 | 5.68 |
| CHEMBL26687 | MESCALINE | 1.0 | 1 | 5.26 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL319415 | — | Ki | = | 2100.0 | nM | 5.68 |
| CHEMBL26687 | MESCALINE | Ki | = | 5500.0 | nM | 5.26 |