Assay Detail
Functional
CHEMBL619029
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Efficient 5-hydroxytryptamine 4 agonist in the rat tunica muscularis mucosae
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Tissue | Muscularis mucosa |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
5-HT4 receptor ligands: applications and new prospects.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 7.51 | 7.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL34291 | — | — | 1 | 7.62 |
| CHEMBL324057 | — | — | 1 | 7.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL34291 | — | EC50 | = | 23.7 | nM | 7.62 |
| CHEMBL324057 | — | EC50 | = | 40.3 | nM | 7.39 |