Assay Detail
Binding
CHEMBL643914
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory activity against Alpha-2 adrenergic receptor in rat vas deferens
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Vas deferens |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Heteroaromatic analogues of the alpha 2-adrenoreceptor partial agonist clonidine.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.11 | 7.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1215 | PHENYLEPHRINE | 4.0 | 1 | 7.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1215 | PHENYLEPHRINE | IC50 | = | 78.0 | nM | 7.11 |