Assay Detail
Binding
CHEMBL652610
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Compound was evaluated for 50% inhibitory concentration against angiotensin II receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
1,4-substituted indoles: a potent and selective class of angiostensin II receptor antagonists
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.53 | 6.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL274447 | — | — | 1 | 6.64 |
| CHEMBL290453 | — | — | 1 | 6.55 |
| CHEMBL27589 | — | — | 1 | 6.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL274447 | — | IC50 | = | 230.0 | nM | 6.64 |
| CHEMBL290453 | — | IC50 | = | 280.0 | nM | 6.55 |
| CHEMBL27589 | — | IC50 | = | 400.0 | nM | 6.40 |