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Assay Detail

CHEMBL652985

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Functional
Antiviral activity was tested using an enzyme-linked immunosorbent assay (ELISA) to detect HSV-1 (herpes simplex virus type 1) using BSC-1 cells
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Cercopithecidae
Cell Type BSC-1
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

ADMET (CHEMBL612558)
Type ADMET

Publication

Deoxy sugar analogues of triciribine: correlation of antiviral and antiproliferative activity with intracellular phosphorylation.
Porcari AR, Ptak RG, Borysko KZ, Breitenbach JM, Vittori S, Wotring LL, Drach JC, Townsend LB.
J Med Chem (2000) 43 : 2438 -2448
PubMed 10882371 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 8 4.69 5.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1790617 1 5.22
CHEMBL462018 TRICIRIBINE PHOSPHATE 2.0 1 4.70
CHEMBL331237 TRICIRIBINE 1 4.64
CHEMBL315509 1 4.19
CHEMBL314567 1 -
CHEMBL2367598 1 -
CHEMBL2112098 1 -
CHEMBL609194 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1790617 IC50 = 6000.0 nM 5.22
CHEMBL462018 TRICIRIBINE PHOSPHATE IC50 = 20000.0 nM 4.70
CHEMBL331237 TRICIRIBINE IC50 = 23000.0 nM 4.64
CHEMBL315509 IC50 = 65000.0 nM 4.19
CHEMBL314567 IC50 > 100000.0 nM -
CHEMBL2367598 IC50 > 100000.0 nM -
CHEMBL2112098 IC50 > 100000.0 nM -
CHEMBL609194 IC50 > 100000.0 nM -