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Assay Detail

CHEMBL663530

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibition of heterologously expressed human cytochrome P450 2D6
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Expert

Target

Cytochrome P450 2D6 (CHEMBL289)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Biarylcarbamoylindolines are novel and selective 5-HT(2C) receptor inverse agonists: identification of 5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a potential antidepressant/anxiolytic agent.
Bromidge SM, Dabbs S, Davies DT, Davies S, Duckworth DM, Forbes IT, Gaster LM, Ham P, Jones GE, King FD, Mulholland KR, Saunders DV, Wyman PA, Blaney FE, Clarke SE, Blackburn TP, Holland V, Kennett GA, Lightowler S, Middlemiss DN, Trail B, Riley GJ, Wood MD.
J Med Chem (2000) 43 : 1123 -1134
PubMed 10737744 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 5.82 6.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL276140 1 6.96
CHEMBL14276 1 4.68
CHEMBL14563 SB-242084 1 -
CHEMBL14460 SB-243213 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL276140 IC50 = 110.0 nM 6.96
CHEMBL14276 IC50 = 21000.0 nM 4.68
CHEMBL14563 SB-242084 IC50 > 100000.0 nM -
CHEMBL14460 SB-243213 IC50 > 100000.0 nM -