Assay Detail
Binding
CHEMBL665832
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Compound was evaluated in an intact RBL-1 cell line for inhibition of 5-Cyclooxygenase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | RBL-1 |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Conversion of NSAIDS into balanced dual inhibitors of cyclooxygenase and 5-lipoxygenase
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.00 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL509 | MECLOFENAMIC ACID | 4.0 | 1 | 7.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL509 | MECLOFENAMIC ACID | IC50 | = | 100.0 | nM | 7.00 |