Assay Detail
Binding
CHEMBL665876
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of the murine Arg120Ala mutant type COX-2
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Amide derivatives of meclofenamic acid as selective cyclooxygenase-2 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.40 | 6.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL509 | MECLOFENAMIC ACID | 4.0 | 1 | 6.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL509 | MECLOFENAMIC ACID | IC50 | = | 400.0 | nM | 6.40 |