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Assay Detail

CHEMBL674318

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Effective concentration required to inhibit Herpes simplex virus-1(HSV-1) / thymine kinase deficient (TK-)B2006 / VMW1837 induced cytopathicity by 50% in E6SM cell lines
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Cell Type E6SM
Confidence 1 — Organism
Curated By Intermediate

Target

E6SM (CHEMBL614149)
Type CELL-LINE
Organism Homo sapiens

Publication

Synthesis, mechanism of action, and antiviral activity of a new series of covalent mechanism-based inhibitors of S-adenosyl-L-homocysteine hydrolase.
Guillerm G, Guillerm D, Vandenplas-Witkowki C, Rogniaux H, Carte N, Leize E, Van Dorsselaer A, De Clercq E, Lambert C.
J Med Chem (2001) 44 : 2743 -2752
PubMed 11495586 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 8.30 8.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1643 RIBAVIRIN 4.0 1 8.30
CHEMBL140440 1 -
CHEMBL607985 1 -
CHEMBL606446 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1643 RIBAVIRIN EC50 = 5.0 nM 8.30
CHEMBL140440 EC50 > 250000.0 nM -
CHEMBL607985 EC50 > 250000.0 nM -
CHEMBL606446 EC50 = 150000.0 nM -