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Assay Detail

CHEMBL675730

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Binding
Compound was evaluated for binding activity against [3H]haloperidol as radioligand for Dopamine receptor D2
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

D(2) dopamine receptor (CHEMBL339)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

In vitro labeling of serotonin-S2 receptors: synthesis and binding characteristics of [3H]-7-aminoketanserin.
Wouters W, Janssen CG, Van Dun J, Thijssen JB, Laduron PM.
J Med Chem (1986) 29 : 1663 -1668
PubMed 3746815 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 6.79 6.79

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL46683 1 6.79

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL46683 Ki = 164.0 nM 6.79