Assay Detail
Binding
CHEMBL680569
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Affinity on glycogen phosphorylase (GP) enzyme.
30
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Three-dimensional quantitative structure-activity relationships from molecular similarity matrices and genetic neural networks. 2. Applications.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 30 | 4.57 | 5.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3351144 | — | — | 1 | 5.52 |
| CHEMBL133097 | — | — | 1 | 4.80 |
| CHEMBL3351143 | — | — | 1 | 4.50 |
| CHEMBL3351132 | — | — | 1 | 4.35 |
| CHEMBL3351152 | — | — | 1 | 4.23 |
| CHEMBL3351139 | — | — | 1 | 4.03 |
| CHEMBL136618 | — | — | 1 | - |
| CHEMBL3351136 | — | — | 1 | - |
| CHEMBL3351153 | — | — | 1 | - |
| CHEMBL3351145 | — | — | 1 | - |
| CHEMBL3351141 | — | — | 1 | - |
| CHEMBL284555 | — | — | 1 | - |
| CHEMBL71477 | — | — | 1 | - |
| CHEMBL334655 | — | — | 2 | - |
| CHEMBL3351150 | — | — | 1 | - |
| CHEMBL335028 | — | — | 1 | - |
| CHEMBL134001 | — | — | 1 | - |
| CHEMBL35946 | — | — | 2 | - |
| CHEMBL1222250 | DEXTROSE | 4.0 | 1 | - |
| CHEMBL3351149 | — | — | 1 | - |
| CHEMBL35563 | — | — | 1 | - |
| CHEMBL3351138 | — | — | 1 | - |
| CHEMBL35757 | — | — | 2 | - |
| CHEMBL3351135 | — | — | 1 | - |
| CHEMBL3215399 | — | — | 1 | - |
| CHEMBL423484 | — | — | 1 | - |
| CHEMBL3351133 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3351144 | — | Ki | = | 2999.16 | nM | 5.52 |
| CHEMBL133097 | — | Ki | = | 15995.58 | nM | 4.80 |
| CHEMBL3351143 | — | Ki | = | 31988.95 | nM | 4.50 |
| CHEMBL3351132 | — | Ki | = | 44977.99 | nM | 4.35 |
| CHEMBL3351152 | — | Ki | = | 59020.11 | nM | 4.23 |
| CHEMBL3351139 | — | Ki | = | 93972.33 | nM | 4.03 |
| CHEMBL35946 | — | Ki | = | 36728230.05 | nM | - |
| CHEMBL136618 | — | Ki | = | 18879913.49 | nM | - |
| CHEMBL134001 | — | Ki | = | 1999861.87 | nM | - |
| CHEMBL3351133 | — | Ki | = | 21086281.5 | nM | - |
| CHEMBL3351150 | — | Ki | = | 369828.18 | nM | - |
| CHEMBL334655 | — | Ki | = | 399944.75 | nM | - |
| CHEMBL71477 | — | Ki | = | 16788040.18 | nM | - |
| CHEMBL284555 | — | Ki | = | 2798981.32 | nM | - |
| CHEMBL3351141 | — | Ki | = | 990831.94 | nM | - |
| CHEMBL3351145 | — | Ki | = | 1300169.58 | nM | - |
| CHEMBL3351153 | — | Ki | = | 145881.43 | nM | - |
| CHEMBL3351136 | — | Ki | = | 1798870.92 | nM | - |
| CHEMBL423484 | — | Ki | = | 4797334.49 | nM | - |
| CHEMBL3215399 | — | Ki | = | 16292960.33 | nM | - |
| CHEMBL35946 | — | Ki | = | 159955.8 | nM | - |
| CHEMBL35757 | — | Ki | = | 369828.18 | nM | - |
| CHEMBL334655 | — | Ki | = | 2999162.52 | nM | - |
| CHEMBL3351135 | — | Ki | = | 3597493.35 | nM | - |
| CHEMBL335028 | — | Ki | = | 15205475.3 | nM | - |
| CHEMBL3351138 | — | Ki | = | 139958.73 | nM | - |
| CHEMBL35563 | — | Ki | = | 5597576.01 | nM | - |
| CHEMBL3351149 | — | Ki | = | 16904409.32 | nM | - |
| CHEMBL1222250 | DEXTROSE | Ki | = | 1698243.65 | nM | - |
| CHEMBL35757 | — | Ki | = | 439541.62 | nM | - |