Assay Detail
Functional
CHEMBL683607
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Opiod agonistic activity against delta enriched smooth muscle preparation
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cavia porcellus |
| Tissue | Muscle tissue |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Opioid agonist and antagonist activities of morphindoles related to naltrindole.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.84 | 6.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL285563 | — | — | 1 | 6.92 |
| CHEMBL607339 | — | — | 1 | 6.76 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL285563 | — | IC50 | = | 121.0 | nM | 6.92 |
| CHEMBL607339 | — | IC50 | = | 174.0 | nM | 6.76 |