Assay Detail
Functional
CHEMBL684566
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Increasing force in skinned fibers at constant buffered Ca-concentration
3
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cavia porcellus |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Preparation of the enantiomers of the novel CA-sensitizer EMD 53 998
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 5.55 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL314612 | — | — | 3 | 5.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL314612 | — | EC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL314612 | — | EC50 | = | 4800.0 | nM | 5.32 |
| CHEMBL314612 | — | EC50 | > | 100000.0 | nM | - |