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Assay Detail

CHEMBL688858

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antioxidative activity was evaluated by using the lipid peroxidation of guinea pig liver microsomes
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Cavia porcellus
Tissue Liver
Subcellular Microsomes
Confidence 1 — Organism
Curated By Intermediate

Target

Cavia porcellus (CHEMBL369)
Type ORGANISM
Organism Cavia porcellus

Publication

Total synthesis of an antioxidant isolated from yeast via palladium-catalyzed coupling and its application for related compounds.
Jinno S, Okita T, Inouye K.
Bioorg Med Chem Lett (1999) 9 : 1029 -1032
PubMed 10230633 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 8 4.20 4.36

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL8115 1 4.36
CHEMBL7983 PROPYL GALLATE 1.0 1 4.30
CHEMBL7998 1 4.25
CHEMBL274614 1 4.19
CHEMBL8174 1 4.08
CHEMBL274615 1 4.01
CHEMBL47 ALPHA-TOCOPHEROL 1 -
CHEMBL267296 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL8115 IC50 = 44000.0 nM 4.36
CHEMBL7983 PROPYL GALLATE IC50 = 50000.0 nM 4.30
CHEMBL7998 IC50 = 56000.0 nM 4.25
CHEMBL274614 IC50 = 65000.0 nM 4.19
CHEMBL8174 IC50 = 83000.0 nM 4.08
CHEMBL274615 IC50 = 98000.0 nM 4.01
CHEMBL47 ALPHA-TOCOPHEROL IC50 = 280000.0 nM -
CHEMBL267296 IC50 = 107000.0 nM -