Assay Detail
Functional
CHEMBL689701
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro potency in reversing vecuronium-induced block in guinea pig hemidiaphram
36
Total Activities
36
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cavia porcellus |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Oxyaniliniums as acetylcholinesterase inhibitors for the reversal of neuromuscular block.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 36 | 5.47 | 7.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL54126 | NEOSTIGMINE BROMIDE | 2.0 | 1 | 7.55 |
| CHEMBL58511 | — | — | 1 | 6.30 |
| CHEMBL60074 | — | — | 1 | 5.77 |
| CHEMBL59790 | — | — | 1 | 5.70 |
| CHEMBL60745 | EDROPHONIUM BROMIDE | — | 1 | 5.56 |
| CHEMBL58194 | — | — | 1 | 5.54 |
| CHEMBL59192 | — | — | 1 | 5.41 |
| CHEMBL300170 | — | — | 1 | 5.39 |
| CHEMBL62031 | — | — | 1 | 5.15 |
| CHEMBL60180 | — | — | 1 | 5.01 |
| CHEMBL61312 | — | — | 1 | 4.89 |
| CHEMBL61965 | — | — | 1 | 4.71 |
| CHEMBL60596 | — | — | 1 | 4.13 |
| CHEMBL294498 | — | — | 1 | - |
| CHEMBL293751 | — | — | 1 | - |
| CHEMBL61905 | — | — | 1 | - |
| CHEMBL59074 | — | — | 1 | - |
| CHEMBL293316 | — | — | 1 | - |
| CHEMBL57842 | — | — | 1 | - |
| CHEMBL299898 | — | — | 1 | - |
| CHEMBL294674 | — | — | 1 | - |
| CHEMBL294292 | — | — | 1 | - |
| CHEMBL59490 | — | — | 1 | - |
| CHEMBL294152 | — | — | 1 | - |
| CHEMBL60874 | — | — | 1 | - |
| CHEMBL305386 | — | — | 1 | - |
| CHEMBL61126 | — | — | 1 | - |
| CHEMBL294897 | — | — | 1 | - |
| CHEMBL58190 | — | — | 1 | - |
| CHEMBL58252 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL54126 | NEOSTIGMINE BROMIDE | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL58511 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL60074 | — | IC50 | = | 1690.0 | nM | 5.77 |
| CHEMBL59790 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL60745 | EDROPHONIUM BROMIDE | IC50 | = | 2770.0 | nM | 5.56 |
| CHEMBL58194 | — | IC50 | = | 2890.0 | nM | 5.54 |
| CHEMBL59192 | — | IC50 | = | 3870.0 | nM | 5.41 |
| CHEMBL300170 | — | IC50 | = | 4110.0 | nM | 5.39 |
| CHEMBL62031 | — | IC50 | = | 7080.0 | nM | 5.15 |
| CHEMBL60180 | — | IC50 | = | 9800.0 | nM | 5.01 |
| CHEMBL61312 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL61965 | — | IC50 | = | 19400.0 | nM | 4.71 |
| CHEMBL60596 | — | IC50 | = | 74000.0 | nM | 4.13 |
| CHEMBL61515 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL442361 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL58034 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL62210 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL57003 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL291783 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL294498 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL293751 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL61905 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL59074 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL293316 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL57842 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL299898 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL294674 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL294292 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL59490 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL294152 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL60874 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL305386 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL61126 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL294897 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL58190 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL58252 | — | IC50 | > | 3000.0 | nM | - |