Assay Detail
Functional
CHEMBL702286
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Inhibitory activity against growth of JURKAT cells after 144h.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Jurkat |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Effect of polyamine analogues on hypusine content in JURKAT T-cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.43 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL77101 | DIETHYLHOMOSPERMINE | 1.0 | 1 | 6.70 |
| CHEMBL34476 | — | — | 1 | 4.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL77101 | DIETHYLHOMOSPERMINE | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL34476 | — | IC50 | = | 70000.0 | nM | 4.16 |