Assay Detail
Functional
CHEMBL702289
Review assay metadata, readout intent, target linkage, and publication context from the same page.
competitive inhibition of [3H]SPD transport by JURKAT cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Jurkat |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Effect of polyamine analogues on hypusine content in JURKAT T-cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 4.85 | 4.86 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL35633 | — | — | 1 | 4.86 |
| CHEMBL44083 | BIS(ETHYL)NORSPERMINE | — | 1 | 4.84 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL35633 | — | Ki | = | 13800.0 | nM | 4.86 |
| CHEMBL44083 | BIS(ETHYL)NORSPERMINE | Ki | = | 14400.0 | nM | 4.84 |