Assay Detail
Binding
CHEMBL704113
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Inhibitory activity against Janus Kinase 3 protein tyrosine kinase.
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Mapping the kinase domain of Janus Kinase 3.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 6.47 | 7.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL104963 | — | — | 1 | 7.58 |
| CHEMBL323994 | — | — | 1 | 7.57 |
| CHEMBL106571 | — | — | 1 | 7.52 |
| CHEMBL106944 | — | — | 1 | 6.78 |
| CHEMBL107166 | — | — | 1 | 6.72 |
| CHEMBL105255 | — | — | 1 | 6.70 |
| CHEMBL421213 | — | — | 1 | 6.68 |
| CHEMBL107225 | — | — | 1 | 6.67 |
| CHEMBL318390 | — | — | 1 | 6.63 |
| CHEMBL106961 | — | — | 1 | 6.58 |
| CHEMBL320646 | — | — | 1 | 6.46 |
| CHEMBL104062 | — | — | 1 | 6.16 |
| CHEMBL87325 | — | — | 1 | 6.15 |
| CHEMBL104409 | — | — | 1 | 6.06 |
| CHEMBL86755 | — | — | 1 | 6.05 |
| CHEMBL321855 | — | — | 1 | 5.64 |
| CHEMBL107273 | — | — | 1 | 5.31 |
| CHEMBL104640 | — | — | 1 | 5.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL104963 | — | IC50 | = | 26.0 | nM | 7.58 |
| CHEMBL323994 | — | IC50 | = | 27.0 | nM | 7.57 |
| CHEMBL106571 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL106944 | — | IC50 | = | 168.0 | nM | 6.78 |
| CHEMBL107166 | — | IC50 | = | 190.0 | nM | 6.72 |
| CHEMBL105255 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL421213 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL107225 | — | IC50 | = | 213.0 | nM | 6.67 |
| CHEMBL318390 | — | IC50 | = | 235.0 | nM | 6.63 |
| CHEMBL106961 | — | IC50 | = | 260.0 | nM | 6.58 |
| CHEMBL320646 | — | IC50 | = | 350.0 | nM | 6.46 |
| CHEMBL104062 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL87325 | — | IC50 | = | 710.0 | nM | 6.15 |
| CHEMBL104409 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL86755 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL321855 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL107273 | — | IC50 | = | 4900.0 | nM | 5.31 |
| CHEMBL104640 | — | IC50 | = | 7100.0 | nM | 5.15 |