Assay Detail
Binding
CHEMBL710991
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Effect of compound on Melatonin receptor in chicken brain in the presence of MnCl2
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Design and synthesis of new naphthalenic derivatives as ligands for 2-[125I]iodomelatonin binding sites.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.75 | 9.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL294517 | — | — | 1 | 9.75 |
| CHEMBL45 | MELATONIN | 4.0 | 1 | 9.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL294517 | — | Ki | = | 0.176 | nM | 9.75 |
| CHEMBL45 | MELATONIN | Ki | = | 0.176 | nM | 9.75 |