Assay Detail
Functional
CHEMBL737751
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro inhibition of electrically induced contractions in isolated mouse vas deferens (MVD) preparations.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
C-Attached aminoalkylindoles: potent cannabinoid mimetics
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.01 | 8.59 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL69593 | — | — | 1 | 8.59 |
| CHEMBL424042 | — | — | 1 | 7.43 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL69593 | — | IC50 | = | 2.6 | nM | 8.59 |
| CHEMBL424042 | — | IC50 | = | 37.0 | nM | 7.43 |