Assay Detail
Binding
CHEMBL747466
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Binding of [3H]QNB to HM1 receptor was evaluated by saturation binding assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
First fatty acylated dipeptides to affect muscarinic receptor ligand binding.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 10.46 | 10.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL112297 | — | — | 1 | 10.52 |
| CHEMBL115078 | — | — | 1 | 10.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL112297 | — | Kd | = | 0.03 | nM | 10.52 |
| CHEMBL115078 | — | Kd | = | 0.04 | nM | 10.40 |