Assay Detail
Binding
CHEMBL747467
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Ability to displace [3H]QNB from HM1 receptor binding to acetylcholine was evaluated by ligand inhibition assay
2
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
First fatty acylated dipeptides to affect muscarinic receptor ligand binding.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.52 | 10.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL112297 | — | — | 2 | 10.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL112297 | — | Ki | = | 0.01288 | nM | 10.89 |
| CHEMBL112297 | — | Ki | = | 707.95 | nM | 6.15 |