Assay Detail
Functional
CHEMBL750216
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of outward potassium currents (IKn) in human T-lymphocyte N-type potassium channels.
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Target
Potassium voltage-gated channel subfamily A member 3 (CHEMBL4633) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Novel inhibitors of potassium ion channels on human T lymphocytes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 6.34 | 6.67 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL416313 | — | — | 1 | 6.67 |
| CHEMBL298622 | — | — | 1 | 6.67 |
| CHEMBL53676 | — | — | 1 | 6.64 |
| CHEMBL54934 | — | — | 1 | 6.60 |
| CHEMBL299668 | — | — | 1 | 6.60 |
| CHEMBL54846 | — | — | 1 | 6.59 |
| CHEMBL293721 | — | — | 1 | 6.57 |
| CHEMBL56590 | — | — | 1 | 6.55 |
| CHEMBL55202 | — | — | 1 | 6.48 |
| CHEMBL53841 | — | — | 1 | 6.47 |
| CHEMBL298608 | — | — | 1 | 6.46 |
| CHEMBL56589 | — | — | 1 | 6.36 |
| CHEMBL59308 | — | — | 1 | 6.22 |
| CHEMBL56173 | — | — | 1 | 5.98 |
| CHEMBL56261 | — | — | 1 | 5.78 |
| CHEMBL293083 | — | — | 1 | 5.58 |
| CHEMBL55791 | — | — | 1 | 5.50 |
| CHEMBL59482 | — | — | 1 | - |
| CHEMBL293719 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL416313 | — | IC50 | = | 213.0 | nM | 6.67 |
| CHEMBL298622 | — | IC50 | = | 216.0 | nM | 6.67 |
| CHEMBL53676 | — | IC50 | = | 231.0 | nM | 6.64 |
| CHEMBL54934 | — | IC50 | = | 249.0 | nM | 6.60 |
| CHEMBL299668 | — | IC50 | = | 250.0 | nM | 6.60 |
| CHEMBL54846 | — | IC50 | = | 259.0 | nM | 6.59 |
| CHEMBL293721 | — | IC50 | = | 267.0 | nM | 6.57 |
| CHEMBL56590 | — | IC50 | = | 279.0 | nM | 6.55 |
| CHEMBL55202 | — | IC50 | = | 329.0 | nM | 6.48 |
| CHEMBL53841 | — | IC50 | = | 335.0 | nM | 6.47 |
| CHEMBL298608 | — | IC50 | = | 351.0 | nM | 6.46 |
| CHEMBL56589 | — | IC50 | = | 434.0 | nM | 6.36 |
| CHEMBL59308 | — | IC50 | = | 602.0 | nM | 6.22 |
| CHEMBL56173 | — | IC50 | = | 1053.0 | nM | 5.98 |
| CHEMBL56261 | — | IC50 | = | 1676.0 | nM | 5.78 |
| CHEMBL293083 | — | IC50 | = | 2620.0 | nM | 5.58 |
| CHEMBL55791 | — | IC50 | = | 3160.0 | nM | 5.50 |
| CHEMBL59482 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL293719 | — | IC50 | > | 10000.0 | nM | - |