Assay Detail
Binding
CHEMBL753996
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Tested for binding activity against delta opioid receptor using [3H]naltridole ligand
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Synthesis of naltrexone-derived delta-opioid antagonists. Role of conformation of the delta address moiety.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 10.33 | 10.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL610293 | — | — | 1 | 10.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL610293 | — | Ki | = | 0.047 | nM | 10.33 |