Assay Detail
Binding
CHEMBL754470
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of [3H]- ]DSLET binding to Opioid receptor delta 1 from rat brain membrane
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Conformationally restricted deltorphin analogues.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 7.91 | 8.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL124435 | — | — | 1 | 8.30 |
| CHEMBL124941 | — | — | 1 | 8.27 |
| CHEMBL337898 | — | — | 1 | 7.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL124435 | — | Ki | = | 4.96 | nM | 8.30 |
| CHEMBL124941 | — | Ki | = | 5.36 | nM | 8.27 |
| CHEMBL337898 | — | Ki | = | 67.2 | nM | 7.17 |