Assay Detail
Binding
CHEMBL754471
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of [3H]- ]DSLET binding to Opioid receptor delta 1 from rat brain membrane
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Conformationally restricted deltorphin analogues.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.14 | 8.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL339089 | — | — | 1 | 8.19 |
| CHEMBL262312 | — | — | 1 | 8.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL339089 | — | Ki | = | 6.49 | nM | 8.19 |
| CHEMBL262312 | — | Ki | = | 8.27 | nM | 8.08 |