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Assay Detail

CHEMBL754899

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
In vitro cytotoxic activity against mouse leukemia (P388 ) cell line
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type P388
Confidence 1 — Organism
Curated By Intermediate

Target

P388 (CHEMBL389)
Type CELL-LINE
Organism Mus musculus

Publication

Structural requirements for biological activity of the marine alkaloid ascididemin
Lindsay BS, Barrows LR, Copp BR
Bioorg Med Chem Lett (1995) 5 : 739 -742
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 5.22 6.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL340160 ASCIDIDEMIN 1 6.40
CHEMBL133514 BENZOSAMPANGINE 1 5.80
CHEMBL129860 1 4.41
CHEMBL162159 1 4.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL340160 ASCIDIDEMIN IC50 = 400.0 nM 6.40
CHEMBL133514 BENZOSAMPANGINE IC50 = 1600.0 nM 5.80
CHEMBL129860 IC50 = 39000.0 nM 4.41
CHEMBL162159 IC50 = 56000.0 nM 4.25