Assay Detail
Functional
CHEMBL755047
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity against phospholipase C coupled human P2Y purinoceptor 11 (P2Y11)
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Purine and pyrimidine (P2) receptors as drug targets.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 10 | 5.02 | 5.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL336292 | — | — | 1 | 5.82 |
| CHEMBL131890 | ATPGAMMAS | — | 1 | 5.52 |
| CHEMBL339386 | — | — | 1 | 5.16 |
| CHEMBL335538 | — | — | 1 | 5.05 |
| CHEMBL14249 | ADENOSINE TRIPHOSPHATE | 2.0 | 1 | 4.77 |
| CHEMBL335206 | — | — | 1 | 4.52 |
| CHEMBL336208 | — | — | 1 | 4.30 |
| CHEMBL336296 | URIDINE TRIPHOSPHATE | 3.0 | 1 | - |
| CHEMBL3085531 | — | — | 1 | - |
| CHEMBL223344 | RB 2 | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL336292 | — | EC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL131890 | ATPGAMMAS | EC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL339386 | — | EC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL335538 | — | EC50 | = | 9000.0 | nM | 5.05 |
| CHEMBL14249 | ADENOSINE TRIPHOSPHATE | EC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL335206 | — | EC50 | = | 30000.0 | nM | 4.52 |
| CHEMBL336208 | — | EC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL336296 | URIDINE TRIPHOSPHATE | EC50 | > | 100000.0 | nM | - |
| CHEMBL3085531 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL223344 | RB 2 | EC50 | > | 100000.0 | nM | - |