Assay Detail
Functional
CHEMBL760183
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Compound was evaluated in rabbit-platelet rich plasma (PRP) for the molar concentration required to produce 50% of maximum aggregation
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Oryctolagus cuniculus |
| Tissue | Plasma |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Analogues of platelet activating factor. 5. Multiple oxygen substitution of the alkoxy chain.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 6.43 | 7.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL17935 | PLATELET ACTIVATING FACTOR | — | 1 | 7.58 |
| CHEMBL416745 | — | — | 1 | 5.28 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL17935 | PLATELET ACTIVATING FACTOR | EC50 | = | 26.5 | nM | 7.58 |
| CHEMBL416745 | — | EC50 | = | 5300.0 | nM | 5.28 |