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Assay Detail

CHEMBL762236

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity for cloned human oxytocin receptor (OT-R)
36
Total Activities
36
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Oxytocin receptor (CHEMBL2049)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Development of orally active oxytocin antagonists: studies on 1-(1-[4-[1-(2-methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl]piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and related pyridines.
Bell IM, Erb JM, Freidinger RM, Gallicchio SN, Guare JP, Guidotti MT, Halpin RA, Hobbs DW, Homnick CF, Kuo MS, Lis EV, Mathre DJ, Michelson SR, Pawluczyk JM, Pettibone DJ, Reiss DR, Vickers S, Williams PD, Woyden CJ.
J Med Chem (1998) 41 : 2146 -2163
PubMed 9622556 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 36 8.38 9.09

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL66985 1 9.09
CHEMBL303700 1 9.09
CHEMBL302297 1 9.00
CHEMBL308673 1 9.00
CHEMBL306416 1 8.96
CHEMBL71540 1 8.92
CHEMBL66931 1 8.85
CHEMBL68480 1 8.82
CHEMBL68800 1 8.77
CHEMBL66992 1 8.70
CHEMBL66240 1 8.68
CHEMBL265070 1 8.64
CHEMBL302128 1 8.64
CHEMBL69202 1 8.60
CHEMBL302029 1 8.60
CHEMBL68816 1 8.48
CHEMBL303487 1 8.46
CHEMBL306645 1 8.39
CHEMBL306010 1 8.38
CHEMBL24781 1 8.32
CHEMBL308460 1 8.32
CHEMBL68199 1 8.29
CHEMBL65949 1 8.28
CHEMBL65950 1 8.25
CHEMBL69265 1 8.17
CHEMBL69201 1 8.15
CHEMBL68978 1 8.11
CHEMBL68914 1 8.00
CHEMBL69539 1 7.96
CHEMBL69520 1 7.96

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL66985 Ki = 0.81 nM 9.09
CHEMBL303700 Ki = 0.82 nM 9.09
CHEMBL308673 Ki = 1.0 nM 9.00
CHEMBL302297 Ki = 1.0 nM 9.00
CHEMBL306416 Ki = 1.1 nM 8.96
CHEMBL71540 Ki = 1.2 nM 8.92
CHEMBL66931 Ki = 1.4 nM 8.85
CHEMBL68480 Ki = 1.5 nM 8.82
CHEMBL68800 Ki = 1.7 nM 8.77
CHEMBL66992 Ki = 2.0 nM 8.70
CHEMBL66240 Ki = 2.1 nM 8.68
CHEMBL265070 Ki = 2.3 nM 8.64
CHEMBL302128 Ki = 2.3 nM 8.64
CHEMBL69202 Ki = 2.5 nM 8.60
CHEMBL302029 Ki = 2.5 nM 8.60
CHEMBL68816 Ki = 3.3 nM 8.48
CHEMBL303487 Ki = 3.5 nM 8.46
CHEMBL306645 Ki = 4.1 nM 8.39
CHEMBL306010 Ki = 4.2 nM 8.38
CHEMBL308460 Ki = 4.8 nM 8.32
CHEMBL24781 Ki = 4.8 nM 8.32
CHEMBL68199 Ki = 5.1 nM 8.29
CHEMBL65949 Ki = 5.3 nM 8.28
CHEMBL65950 Ki = 5.6 nM 8.25
CHEMBL69265 Ki = 6.7 nM 8.17
CHEMBL69201 Ki = 7.0 nM 8.15
CHEMBL68978 Ki = 7.8 nM 8.11
CHEMBL68914 Ki = 10.0 nM 8.00
CHEMBL69539 Ki = 11.0 nM 7.96
CHEMBL69520 Ki = 11.0 nM 7.96
CHEMBL68752 Ki = 13.0 nM 7.89
CHEMBL68373 Ki = 14.0 nM 7.85
CHEMBL66749 Ki = 16.0 nM 7.80
CHEMBL66567 Ki = 23.0 nM 7.64
CHEMBL304577 Ki = 29.0 nM 7.54
CHEMBL69498 Ki = 82.0 nM 7.09