Assay Detail
Binding
CHEMBL767411
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Inhibition of protein kinase C gamma
3
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
New hexahydroxybiphenyl derivatives as inhibitors of protein kinase C.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.43 | 4.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL294037 | — | — | 2 | 4.52 |
| CHEMBL59451 | — | — | 1 | 4.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL294037 | — | IC50 | = | 30000.0 | nM | 4.52 |
| CHEMBL294037 | — | IC50 | = | 34000.0 | nM | 4.47 |
| CHEMBL59451 | — | IC50 | = | 50000.0 | nM | 4.30 |