Assay Detail
Binding
CHEMBL769172
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Inhibition of protein kinase C
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
The synthesis and evaluation of diacylglycerol analogues as potential second-messenger antagonists
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.67 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL24609 | MONOCTANOIN COMPONENT C | -1.0 | 1 | 5.00 |
| CHEMBL26341 | — | — | 1 | 5.00 |
| CHEMBL26440 | — | — | 1 | 4.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL24609 | MONOCTANOIN COMPONENT C | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL26341 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL26440 | — | IC50 | = | 100000.0 | nM | 4.00 |