Assay Detail
Binding
CHEMBL769343
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Binding to PKC in 3[H]-PBDU assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Target
Protein kinase C, PKC; classical/novel (CHEMBL2096620) ↗| Type | PROTEIN FAMILY |
| Organism | Homo sapiens |
Publication
Synthesis and biological activity of a 5,6-substituted teleocidin
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.61 | 6.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL120645 | — | — | 1 | 6.82 |
| CHEMBL143453 | — | — | 1 | 6.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL120645 | — | IC50 | = | 150.0 | nM | 6.82 |
| CHEMBL143453 | — | IC50 | = | 400.0 | nM | 6.40 |