Assay Detail
Binding
CHEMBL772954
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human Protein kinase C gamma
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Ring size effect in the PKC inhibitory activities of perhydroazepine analogs of balanol
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.35 | 7.47 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL60254 | BALANOL | — | 1 | 7.47 |
| CHEMBL304549 | — | — | 1 | 7.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL60254 | BALANOL | IC50 | = | 34.0 | nM | 7.47 |
| CHEMBL304549 | — | IC50 | = | 60.0 | nM | 7.22 |