Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL772957

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity for human Protein kinase C gamma with [Ca2+]
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Expert

Target

Protein kinase C gamma type (CHEMBL2938)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

New bivalent PKC ligands linked by a carbon spacer: enhancement in binding affinity.
Sridhar J, Wei ZL, Nowak I, Lewin NE, Ayres JA, Pearce LV, Blumberg PM, Kozikowski AP.
J Med Chem (2003) 46 : 4196 -4204
PubMed 12954072 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 9.80 9.80

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL337834 1 9.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL337834 Kd = 0.16 nM 9.80