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Assay Detail

CHEMBL804696

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Binding
Ability to inhibit [3H]paroxetine binding to cloned human serotonin (5-HT) transporter
9
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Expert

Target

Sodium-dependent serotonin transporter (CHEMBL228)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Synthesis and biological activity of some known and putative duloxetine metabolites.
Kuo F, Gillespie TA, Kulanthaivel P, Lantz RJ, Ma TW, Nelson DL, Threlkeld PG, Wheeler WJ, Yi P, Zmijewski M.
Bioorg Med Chem Lett (2004) 14 : 3481 -3486
PubMed 15177457 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 9 6.91 9.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1175 DULOXETINE 4.0 1 9.10
CHEMBL326713 2 7.50
CHEMBL119605 1 6.58
CHEMBL2029052 1 5.84
CHEMBL420142 1 5.51
CHEMBL2029054 1 -
CHEMBL2029055 1 -
CHEMBL2029053 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1175 DULOXETINE Ki = 0.79 nM 9.10
CHEMBL326713 Ki = 31.7 nM 7.50
CHEMBL326713 Ki = 120.0 nM 6.92
CHEMBL119605 Ki = 266.0 nM 6.58
CHEMBL2029052 Ki = 1459.0 nM 5.84
CHEMBL420142 Ki = 3118.0 nM 5.51
CHEMBL2029054 Ki > 10000.0 nM -
CHEMBL2029055 Ki > 10000.0 nM -
CHEMBL2029053 Ki > 10000.0 nM -