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Assay Detail

CHEMBL812899

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
In Vitro Growth Inhibitory Value against K243 Strain of Trypanosoma brucei.
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Trypanosoma brucei
Confidence 1 — Organism
Curated By Intermediate

Target

Trypanosoma brucei (CHEMBL612849)
Type ORGANISM
Organism Trypanosoma brucei

Publication

Terminally alkylated polyamine analogues as chemotherapeutic agents.
Casero RA, Woster PM.
J Med Chem (2001) 44 : 1 -26
PubMed 11141084 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.40 6.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL313792 MELARSEN OXIDE -1.0 1 6.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL313792 MELARSEN OXIDE IC50 = 400.0 nM 6.40