Assay Detail
Functional
CHEMBL815467
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In vitro growth Inhibitory activity against K269 Strain of Trypanosoma brucei.
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Trypanosoma brucei |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Terminally alkylated polyamine analogues as chemotherapeutic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 5.39 | 6.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL41629 | — | — | 1 | 6.16 |
| CHEMBL289450 | — | — | 1 | 6.12 |
| CHEMBL43390 | — | — | 1 | 5.77 |
| CHEMBL296119 | — | — | 1 | 5.29 |
| CHEMBL40258 | — | — | 1 | 4.91 |
| CHEMBL86435 | — | — | 1 | 4.78 |
| CHEMBL416078 | — | — | 1 | 4.68 |
| CHEMBL86940 | — | — | 1 | - |
| CHEMBL447829 | — | — | 1 | - |
| CHEMBL44039 | — | — | 1 | - |
| CHEMBL33387 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL41629 | — | IC50 | = | 690.0 | nM | 6.16 |
| CHEMBL289450 | — | IC50 | = | 750.0 | nM | 6.12 |
| CHEMBL43390 | — | IC50 | = | 1710.0 | nM | 5.77 |
| CHEMBL296119 | — | IC50 | = | 5100.0 | nM | 5.29 |
| CHEMBL40258 | — | IC50 | = | 12300.0 | nM | 4.91 |
| CHEMBL86435 | — | IC50 | = | 16500.0 | nM | 4.78 |
| CHEMBL416078 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL86940 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL447829 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL44039 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL33387 | — | IC50 | > | 100000.0 | nM | - |