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Assay Detail

CHEMBL817404

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
In vitro growth inhibition of bloodstream-form Trypanosoma brucei rhodesiense Trypomastigotes
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Trypanosoma brucei rhodesiense
Confidence 1 — Organism
Curated By Expert

Target

Trypanosoma brucei rhodesiense (CHEMBL612348)
Type ORGANISM
Organism Trypanosoma brucei rhodesiense

Publication

Activity of bisphosphonates against Trypanosoma brucei rhodesiense.
Martin MB, Sanders JM, Kendrick H, de Luca-Fradley K, Lewis JC, Grimley JS, Van Brussel EM, Olsen JR, Meints GA, Burzynska A, Kafarski P, Croft SL, Oldfield E.
J Med Chem (2002) 45 : 2904 -2914
PubMed 12086478 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 27 5.01 6.66

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL434024 1 6.66
CHEMBL55557 1 6.21
CHEMBL55140 1 6.16
CHEMBL997 IBANDRONIC ACID 4.0 1 6.02
CHEMBL293522 1 5.77
CHEMBL52251 (OCTYLAMINO)METHYLENEDIPHOSPHONIC ACID 1 5.77
CHEMBL416301 1 5.70
CHEMBL55812 OLPADRONIC ACID 2.0 1 5.27
CHEMBL55358 1 5.11
CHEMBL298852 1 5.10
CHEMBL923 RISEDRONIC ACID 4.0 1 5.07
CHEMBL301247 1 5.07
CHEMBL55359 1 4.70
CHEMBL54004 1 4.69
CHEMBL56253 (CYCLOHEXYLAMINO)METHYLENEDIPHOSPHONIC ACID 1 4.68
CHEMBL56556 1 4.67
CHEMBL55214 NERIDRONIC ACID 3.0 1 4.50
CHEMBL54344 (DIETHYLAMINO)METHYLENEDIPHOSPHONIC ACID 1 4.46
CHEMBL417932 1 4.40
CHEMBL100483 1 4.40
CHEMBL56255 (PENTYLAMINO)METHYLENEDIPHOSPHONIC ACID 1 4.30
CHEMBL54714 1 4.27
CHEMBL299988 1 4.21
CHEMBL52761 1 4.04
CHEMBL299491 1 4.00
CHEMBL834 PAMIDRONIC ACID 4.0 1 -
CHEMBL55856 (ISOPENTYLAMINO)METHYLENEDIPHOSPHONIC ACID 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL434024 IC50 = 220.0 nM 6.66
CHEMBL55557 IC50 = 610.0 nM 6.21
CHEMBL55140 IC50 = 700.0 nM 6.16
CHEMBL997 IBANDRONIC ACID IC50 = 960.0 nM 6.02
CHEMBL293522 IC50 = 1700.0 nM 5.77
CHEMBL52251 (OCTYLAMINO)METHYLENEDIPHOSPHONIC ACID IC50 = 1700.0 nM 5.77
CHEMBL416301 IC50 = 2000.0 nM 5.70
CHEMBL55812 OLPADRONIC ACID IC50 = 5400.0 nM 5.27
CHEMBL55358 IC50 = 7800.0 nM 5.11
CHEMBL298852 IC50 = 8000.0 nM 5.10
CHEMBL923 RISEDRONIC ACID IC50 = 8600.0 nM 5.07
CHEMBL301247 IC50 = 8600.0 nM 5.07
CHEMBL55359 IC50 = 19800.0 nM 4.70
CHEMBL54004 IC50 = 20500.0 nM 4.69
CHEMBL56253 (CYCLOHEXYLAMINO)METHYLENEDIPHOSPHONIC ACID IC50 = 20900.0 nM 4.68
CHEMBL56556 IC50 = 21300.0 nM 4.67
CHEMBL55214 NERIDRONIC ACID IC50 = 31700.0 nM 4.50
CHEMBL54344 (DIETHYLAMINO)METHYLENEDIPHOSPHONIC ACID IC50 = 34400.0 nM 4.46
CHEMBL417932 IC50 = 40000.0 nM 4.40
CHEMBL100483 IC50 = 39500.0 nM 4.40
CHEMBL56255 (PENTYLAMINO)METHYLENEDIPHOSPHONIC ACID IC50 = 50600.0 nM 4.30
CHEMBL54714 IC50 = 53300.0 nM 4.27
CHEMBL299988 IC50 = 62400.0 nM 4.21
CHEMBL52761 IC50 = 92000.0 nM 4.04
CHEMBL299491 IC50 = 99800.0 nM 4.00
CHEMBL834 PAMIDRONIC ACID IC50 > 100000.0 nM -
CHEMBL55856 (ISOPENTYLAMINO)METHYLENEDIPHOSPHONIC ACID IC50 = 102000.0 nM -