Assay Detail
Binding
CHEMBL819590
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Compound was evaluated for its inhibitory activity against CO(cyclooxygenase)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Synthesis and cyclooxygenase and 5-lipoxygenase inhibitory activity of some thiazolidene-4-one analogs of meclofenamic acid
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.11 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL509 | MECLOFENAMIC ACID | 4.0 | 1 | 7.00 |
| CHEMBL162840 | — | — | 1 | 5.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL509 | MECLOFENAMIC ACID | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL162840 | — | IC50 | = | 6000.0 | nM | 5.22 |