Assay Detail

CHEMBL821962

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Functional

Charecterization of agonist response of ligand in mouse stomach bioassay measured as affinity of L-365260

ChEMBL ↗

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Target

Mus musculus (CHEMBL375) ↗

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Primary target Mus musculus

CHEMBL375

Anchored from Assay target.

Protein identity Mus musculus

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Functional
Organism	Mus musculus
Tissue	Stomach
Confidence	1 — Organism
Curated By	Intermediate

Target

Mus musculus (CHEMBL375) ↗

Type	ORGANISM
Organism	Mus musculus

Publication

Nonpeptide cholecystokinin-2 receptor agonists.

Kalindjian SB, Dunstone DJ, Low CM, Pether MJ, Roberts SP, Tozer MJ, Watt GF, Shankley NP.
J Med Chem (2001) 44 : 1125 -1133
PubMed 11312913 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
Kd	1	8.01	8.01

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL1328	PENTAGASTRIN	4.0	1	8.01

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL1328	PENTAGASTRIN	Kd	=	9.772	nM	8.01