Assay Detail
Binding
CHEMBL829479
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Inhibitory concentration against [3H]-DHT binding to human sex hormone-binding globulin (SHBG)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Successful in silico discovery of novel nonsteroidal ligands for human sex hormone binding globulin.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.76 | 4.87 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL193200 | — | — | 1 | 4.87 |
| CHEMBL194392 | — | — | 1 | 4.65 |
| CHEMBL195765 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL193200 | — | IC50 | = | 13600.0 | nM | 4.87 |
| CHEMBL194392 | — | IC50 | = | 22400.0 | nM | 4.65 |
| CHEMBL195765 | — | IC50 | = | 124500.0 | nM | - |