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Assay Detail

CHEMBL830895

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibitory activity against cytochrome P450 determined using human liver microsome upon 15 min incubation with probes substrates Tolbutamide (2C9)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Tissue Liver
Subcellular Microsome
Confidence 9 — Direct single protein target
Curated By Expert

Target

Cytochrome P450 2C9 (CHEMBL3397)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Design of bivalent ligands using hydrogen bond linkers: synthesis and evaluation of inhibitors for human beta-tryptase.
Vaz RJ, Gao Z, Pribish J, Chen X, Levell J, Davis L, Albert E, Brollo M, Ugolini A, Cramer DM, Cairns J, Sides K, Liu F, Kwong J, Kang J, Rebello S, Elliot M, Lim H, Chellaraj V, Singleton RW, Li Y.
Bioorg Med Chem Lett (2004) 14 : 6053 -6056
PubMed 15546728 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 5.80 6.32

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL186730 1 6.32
CHEMBL365062 1 5.27
CHEMBL188068 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL186730 IC50 = 480.0 nM 6.32
CHEMBL365062 IC50 = 5380.0 nM 5.27
CHEMBL188068 IC50 > 50000.0 nM -