Assay Detail
Functional
CHEMBL841435
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of ADP-induced platelet in rabbit platelet rich plasma
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Oryctolagus cuniculus |
| Tissue | Plasma |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
1,3-Dihydro-2H-imidazo[4,5-b]quinolin-2-ones--inhibitors of blood platelet cAMP phosphodiesterase and induced aggregation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 5.98 | 6.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL98738 | — | — | 1 | 6.12 |
| CHEMBL99474 | — | — | 1 | 5.83 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL98738 | — | EC50 | = | 750.0 | nM | 6.12 |
| CHEMBL99474 | — | EC50 | = | 1480.0 | nM | 5.83 |