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Assay Detail

CHEMBL841897

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
The compound was tested for inhibition against methacholine induced tonic contraction in guinea pig ileum.
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Cavia porcellus
Tissue Ileum
Confidence 1 — Organism
Curated By Intermediate

Target

Cavia porcellus (CHEMBL369)
Type ORGANISM
Organism Cavia porcellus

Publication

Synthesis, molecular modeling studies, and muscarinic receptor activity of azaprophen analogues.
Triggle DJ, Kwon YW, Abraham P, Pitner JB, Mascarella SW, Carroll FI.
J Med Chem (1991) 34 : 3164 -3171
PubMed 1956033 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 8.25 8.25

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL322582 1 8.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL322582 Kd = 5.623 nM 8.25