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Assay Detail

CHEMBL855307

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Functional
Cytotoxicity against human Jurkat cells
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type Jurkat
Confidence 1 — Organism
Curated By Expert

Target

Jurkat (CHEMBL397)
Type CELL-LINE
Organism Homo sapiens

Publication

Discovery of a novel series of inhibitors of human cytomegalovirus primase.
Cushing TD, Adrian J, Chen X, DiMaio H, Doughan B, Flygare J, Liang L, Mayorga V, Miao S, Mellon H, Peterson MG, Powers JP, Spector F, Stein C, Wright M, Xu D, Ye Q, Jaen J.
Bioorg Med Chem Lett (2006) 16 : 4879 -4883
PubMed 16814545 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.18 4.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL385536 1 4.60
CHEMBL385412 1 4.10
CHEMBL5314375 CIDOFOVIR 4.0 1 4.00
CHEMBL215727 1 4.00
CHEMBL182 GANCICLOVIR 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL385536 IC50 = 25000.0 nM 4.60
CHEMBL385412 IC50 = 80000.0 nM 4.10
CHEMBL5314375 CIDOFOVIR IC50 = 100000.0 nM 4.00
CHEMBL215727 IC50 = 100000.0 nM 4.00
CHEMBL182 GANCICLOVIR IC50 > 100000.0 nM -