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Assay Detail

CHEMBL862304

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of serotonin re-uptake at human serotonin transporter expressed in HEK293 cells
40
Total Activities
40
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type HEK293
Confidence 9 — Direct single protein target
Curated By Expert

Target

Sodium-dependent serotonin transporter (CHEMBL228)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Designing rapid onset selective serotonin re-uptake inhibitors. Part 1: Structure-activity relationships of substituted (1S,4S)-4-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydro-1-naphthaleneamine.
Middleton DS, Andrews M, Glossop P, Gymer G, Jessiman A, Johnson PS, Mackenny M, Pitcher MJ, Rooker T, Stobie A, Tang K, Morgan P.
Bioorg Med Chem Lett (2006) 16 : 1434 -1439
PubMed 16314097 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 40 7.91 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL206697 1 9.00
CHEMBL383706 1 9.00
CHEMBL411693 1 8.70
CHEMBL438257 1 8.70
CHEMBL382810 1 8.70
CHEMBL809 SERTRALINE 4.0 1 8.52
CHEMBL203741 1 8.52
CHEMBL378379 1 8.52
CHEMBL381792 1 8.52
CHEMBL383427 1 8.40
CHEMBL381754 1 8.30
CHEMBL439337 1 8.30
CHEMBL203776 1 8.30
CHEMBL380758 1 8.30
CHEMBL206649 1 8.22
CHEMBL206211 1 8.22
CHEMBL204285 1 8.22
CHEMBL205505 1 8.15
CHEMBL382241 1 8.15
CHEMBL205837 1 8.10
CHEMBL380523 1 8.05
CHEMBL203674 1 8.00
CHEMBL206598 1 8.00
CHEMBL383081 1 7.89
CHEMBL202907 1 7.62
CHEMBL206599 1 7.60
CHEMBL382673 1 7.60
CHEMBL378804 1 7.52
CHEMBL206404 1 7.51
CHEMBL204005 1 7.51

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL206697 IC50 = 1.0 nM 9.00
CHEMBL383706 IC50 = 1.0 nM 9.00
CHEMBL438257 IC50 = 2.0 nM 8.70
CHEMBL382810 IC50 = 2.0 nM 8.70
CHEMBL411693 IC50 = 2.0 nM 8.70
CHEMBL809 SERTRALINE IC50 = 3.0 nM 8.52
CHEMBL203741 IC50 = 3.0 nM 8.52
CHEMBL378379 IC50 = 3.0 nM 8.52
CHEMBL381792 IC50 = 3.0 nM 8.52
CHEMBL383427 IC50 = 4.0 nM 8.40
CHEMBL439337 IC50 = 5.0 nM 8.30
CHEMBL380758 IC50 = 5.0 nM 8.30
CHEMBL203776 IC50 = 5.0 nM 8.30
CHEMBL381754 IC50 = 5.0 nM 8.30
CHEMBL204285 IC50 = 6.0 nM 8.22
CHEMBL206649 IC50 = 6.0 nM 8.22
CHEMBL206211 IC50 = 6.0 nM 8.22
CHEMBL205505 IC50 = 7.0 nM 8.15
CHEMBL382241 IC50 = 7.0 nM 8.15
CHEMBL205837 IC50 = 8.0 nM 8.10
CHEMBL380523 IC50 = 9.0 nM 8.05
CHEMBL206598 IC50 = 10.0 nM 8.00
CHEMBL203674 IC50 = 10.0 nM 8.00
CHEMBL383081 IC50 = 13.0 nM 7.89
CHEMBL202907 IC50 = 24.0 nM 7.62
CHEMBL206599 IC50 = 25.0 nM 7.60
CHEMBL382673 IC50 = 25.0 nM 7.60
CHEMBL378804 IC50 = 30.0 nM 7.52
CHEMBL206404 IC50 = 31.0 nM 7.51
CHEMBL204005 IC50 = 31.0 nM 7.51
CHEMBL203453 IC50 = 54.0 nM 7.27
CHEMBL202910 IC50 = 60.0 nM 7.22
CHEMBL381315 IC50 = 65.0 nM 7.19
CHEMBL203236 IC50 = 70.0 nM 7.16
CHEMBL202755 IC50 = 90.0 nM 7.05
CHEMBL383128 IC50 = 140.0 nM 6.85
CHEMBL203331 IC50 = 240.0 nM 6.62
CHEMBL204323 IC50 = 290.0 nM 6.54
CHEMBL202810 IC50 = 340.0 nM 6.47
CHEMBL381331 IC50 > 1000.0 nM -